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Bioactive Products
Inhibitors Compound Library
A unique collection of 267 Inhibitor natural compounds
Catalog No: Bb221 Inhibitors Compound Library
Screening Details
Size: 1mg/well * 267 Compounds
2mg/well * 267 Compounds
Cat. No. Information
CFN97061 Deoxycalyciphylline B

Deoxycalyciphylline B exhibits hepatic toxicity. Deoxycalyciphylline B and Methyl homosecodaphniphyllate show different inhibitory effects on thephenoloxidase (PO) of Spodoptera exigua (Hbner) and the inhibitor concentrations leading to 50% (IC50) activity lost are estimated to be 2.439 mmol.L-1 for deoxycalyciphyllineB and 0.879mmol.L-1 for methyl homosecodaphniphyllate,respectively.
CFN97067 epsilon-Viniferin

Epsilon-Viniferin is a bacteriostatic stilbenoid as it antagonized the bactericidal activity of vancomycin. Epsilon-viniferin shows a human cytochrome P450 enzymes inhition activity, it exhibits good antioxidant capacity in the DMSO/O(-)(2) polar system (IC50= 0.14 mM). Epsilon-viniferin and epsilon-viniferin pentaacetate slightly reduce cell proliferation but might protect from cell degenerescence.(-)-Trans-epsilon-viniferin is an inhibitor of noradrenaline and 5-hydroxytryptamine uptake and of monoamine oxidase activity, it may be of value as a structural template for the design and development of new antidepressant drugs.
CFN97068 alpha-Viniferin

Alpha-viniferin is a prostaglandin H2 synthase inhibitor, which has anti-inflammatory, anti-oxidant, anti-arthritis, and anti-tumor activities. Alpha-Viniferin inhibits AChE activity is specific, reversible and noncompetitive, in a dose-dependent manner, and the IC50 values of alpha-Viniferin were 2.0 microM. Alpha-Viniferin exhibits a dose-dependent inhibition on cyclooxygenase activity, where 50% of inhibition (IC50) was shown at a final concentration of about 7 microM, it down-regulates STAT-1-inducible inflammatory genes via inhibiting ERK-mediated STAT-1 activation in IFN-gamma-stimulated macrophages.
CFN97075 Alboctalol

Alboctalol inhibits mushroom tyrosinase activity.
CFN90130 Calebassine

Calebassine is a competitive neuromuscular blocking agent, it is also a Mdm2/MdmX inhibitor.